PDE5 inhibitor powder hydroxythiohomosildenafil 139755-85-4
What is Hydroxyhomosildenafil？
Hydroxyhomosildenafil, also known as Lodenafil, is a drug belonging to a class of drugs called PDE5 inhibitor, which many other erectile dysfunction drugs such as sildenafil, tadalafil, and vardenafil also belong to. Like udenafil and avanafil it belongs to a new generation of PDE5 inhibitors.Lodenafil is formulated as a prodrug in the form of the carbonate ester dimer, lodenafil carbonate, which breaks down in the body to form two molecules of the active drug lodenafil. This formulation has higher oral bioavailability than the parent drug.
Hydroxyhomosildenafil Specifications
Product Name
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Chemical Name
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Hydroxyhomosildenafil;5-[2-Ethoxy-5-[[4-(2-hydroxyethyl)-1-piperazinyl]sulfonyl]phenyl]-1,6-dihydro-1-Methyl-3-propyl-7H-pyrazolo[4,3-d]pyriMidin-7-one;Lodenafil
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Brand Name
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Lodenafil, Helleva
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Drug Class
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Aromatics;Drug Analogues;Heterocycles;Sulfur & Selenium Compounds
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CAS Number
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139755-85-4
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InChIKey
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NEYKRKVLEWKOBI-UHFFFAOYSA-N
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Molecular Formula
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C23H32N6O5S
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Molecular Weight
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504.606
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Monoisotopic Mass
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504.215 g/mol
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Melting Point
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183 -185 °C
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Freezing Point
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183 -185 °C
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Biological Half-Life
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N/A
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Color
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Pale Yellow Solid, off white
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Solubility
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Soluble in DMSO
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Storage Temperature
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Refrigerator
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Application
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Enhances male sexual function
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